PCPEP |
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1-(1-phenylcyclopentyl)piperidine
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| CAS Number | |
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| Formula | C16H23N |
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| Molar mass | 229.367 g·mol−1 |
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| 3D model (JSmol) | |
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C1CCN(CC1)C2(CCCC2)C3=CC=CC=C3
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InChI=1S/C16H23N/c1-3-9-15(10-4-1)16(11-5-6-12-16)17-13-7-2-8-14-17/h1,3-4,9-10H,2,5-8,11-14H2 Key:KNZVHCGBSJFKIX-UHFFFAOYSA-N
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PCPEP (1-phenyl-1-piperidinylcyclopentane) is a designer drug from the arylcyclohexylamine family, which has dissociative effects. It is the ring-contracted cyclopentyl homologue of PCP and has around 1/10th the potency of PCP, making it a similar potency to ketamine.[1][2] It has been sold as an illicit drug in Japan.
See also
References
- ^ Shulgin AT, Mac Lean DE (1976). "Illicit synthesis of phencyclidine (PCP) and several of its analogs". Clinical Toxicology. 9 (4): 553–560. doi:10.3109/15563657608988157. PMID 975751.
- ^ Shannon HE, McQuinn RL, Vaupel DB, Cone EJ (February 1983). "Effects of cycloalkyl ring analogs of phencyclidine on behavior in rodents". The Journal of Pharmacology and Experimental Therapeutics. 224 (2): 327–333. doi:10.1016/S0022-3565(25)33474-9. PMID 6822958.
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| AMPARTooltip α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor | |
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| KARTooltip Kainate receptor | |
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| NMDARTooltip N-Methyl-D-aspartate receptor | |
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- See also: Receptor/signaling modulators
- Metabotropic glutamate receptor modulators
- Glutamate metabolism/transport modulators
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| Group I | | mGluR1Tooltip Metabotropic glutamate receptor 1 | |
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| mGluR5Tooltip Metabotropic glutamate receptor 5 | |
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| Group II | | mGluR2Tooltip Metabotropic glutamate receptor 2 | |
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| mGluR3Tooltip Metabotropic glutamate receptor 3 | |
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| Group III | | mGluR4Tooltip Metabotropic glutamate receptor 4 |
- Antagonists: CPPG
- MAP4
- MPPG
- MSOP
- MTPG
- UBP-1112
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| mGluR6Tooltip Metabotropic glutamate receptor 6 |
- Antagonists: CPPG
- MAP4
- MPPG
- MSOP
- MTPG
- UBP-1112
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| mGluR7Tooltip Metabotropic glutamate receptor 7 |
- Antagonists: CPPG
- MAP4
- MMPIP
- MPPG
- MSOP
- MTPG
- UBP-1112
- XAP044; Negative allosteric modulators: ADX71743
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| mGluR8Tooltip Metabotropic glutamate receptor 8 |
- Antagonists: CPPG
- MAP4
- MPPG
- MSOP
- MTPG
- UBP-1112
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See also: Receptor/signaling modulators • Ionotropic glutamate receptor modulators • Glutamate metabolism/transport modulators |
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